Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50023543
Affinity DataKd: 4.40nMAssay Description:Binding affinity to N-terminal His-tagged human RARalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by IT...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at Gal4-fused full length human RARgamma LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at Gal4-fused full length human RARalpha LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataEC50: 16nMAssay Description:Agonist activity at Gal4-fused full length human RARalpha LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataKd: 98nMAssay Description:Binding affinity to N-terminal His-tagged human RARalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataEC50: 419nMAssay Description:Agonist activity at Gal4-fused full length human RARalpha LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataEC50: 424nMAssay Description:Agonist activity at Gal4-fused full length human RARalpha LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataKd: 433nMAssay Description:Binding affinity to N-terminal His-tagged human RARalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Partial agonist activity at Gal4-fused full length RXRalpha LBD (unknown origin) transfected in HEK293T cells co-transfected with pG5luc reporter and...More data for this Ligand-Target Pair
Affinity DataKd: 549nMAssay Description:Binding affinity to N-terminal His-tagged human RXRalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataKd: 553nMAssay Description:Binding affinity to N-terminal His-tagged human RARalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataKd: 663nMAssay Description:Binding affinity to N-terminal His-tagged human RXRalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataIC50: 832nMAssay Description:Partial agonist activity at Gal4-fused full length RXRalpha LBD (unknown origin) transfected in HEK293T cells co-transfected with pG5luc reporter and...More data for this Ligand-Target Pair
Affinity DataKd: 852nMAssay Description:Binding affinity to N-terminal His-tagged human RXRalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fl...More data for this Ligand-Target Pair
Affinity DataEC50: 984nMAssay Description:Agonist activity at Gal4-fused full length human RARbeta LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assesse...More data for this Ligand-Target Pair
Affinity DataKd: 1.08E+3nMAssay Description:Binding affinity to N-terminal His-tagged human RARalpha LBD extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by IT...More data for this Ligand-Target Pair
Affinity DataEC50: 1.14E+3nMAssay Description:Agonist activity at Gal4-fused full length human RARgamma LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataEC50: 2.24E+3nMAssay Description:Agonist activity at Gal4-fused full length human RARgamma LBD transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla-luc assess...More data for this Ligand-Target Pair
Affinity DataEC50: 3.52E+3nMAssay Description:Agonist activity at Gal4-fused full length RXRalpha LBD (unknown origin) transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla...More data for this Ligand-Target Pair
Affinity DataEC50: 4.64E+3nMAssay Description:Agonist activity at Gal4-fused full length RXRalpha LBD (unknown origin) transfected in HEK293T cells co-transfected with pG5luc reporter and Renilla...More data for this Ligand-Target Pair
