Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50022943
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656426BDBM50656426(AT-1 | AT1 | BRD4 DEGRADER AT1 | CHEMBL4455124)
Affinity DataKd:  4.40nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365463BDBM50365463(CHEMBL1232461)
Affinity DataIC50: 33nMAssay Description:Inhibition of His-tagged BRD4 BD1 (144 to 168 residues) (unknown origin) extracted from Escherichia coli using biotinylated histone peptide H4 SGRG-K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365463BDBM50365463(CHEMBL1232461)
Affinity DataKd:  51nMAssay Description:Binding affinity to His-tagged BRD4 BD1 (144 to 168 residues) (unknown origin) extracted from Escherichia coli assessed as dissociation constant by S...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656425BDBM50656425(CHEMBL6162291)
Affinity DataKd:  100nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed