Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50022943
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
Affinity DataKd: 4.40nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of His-tagged BRD4 BD1 (144 to 168 residues) (unknown origin) extracted from Escherichia coli using biotinylated histone peptide H4 SGRG-K...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
Affinity DataKd: 51nMAssay Description:Binding affinity to His-tagged BRD4 BD1 (144 to 168 residues) (unknown origin) extracted from Escherichia coli assessed as dissociation constant by S...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
National Institute of Science Education and Research (NISER)
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair


