Report error Found 293 Enz. Inhib. hit(s) with all data for entry = 50022955
Affinity DataKi: 10nMAssay Description:Binding affinity to SARS-CoV-2 Main protease assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 Main protease assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 Main protease assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 Main protease assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of SARS-CoV-2 3CL protease extracted from Escherichia coli BL21 (DE3) Rosetta cells using DabcylKNSTLQSGLRKE-Edan as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease (PLpro) by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease (PLpro) by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease (PLpro) by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease (PLpro) by enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity to SARS-CoV-2 papain-like protease extracted from Escherichia coli BL21 (DE3) cells assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 papain-like proteaseMore data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease extracted from Escherichia coli BL21 (DE3) Rosetta cells assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 3CL protease by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of SARS-CoV-2 Main protease using Dabcyl-KLSAVLQSGFRKM-Edans-NH2 as substrate incubated for 30 mins by by FRET based enzymatic assayMore data for this Ligand-Target Pair















































