Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50022977
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657136BDBM50657136(CHEMBL6147947)
Affinity DataEC50:  1.40nMAssay Description:Activation of KV7.2/3 channel transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657113BDBM50657113(CHEMBL6147914)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81199BDBM81199((Z)-but-2-enedioate;ethyl N-[2-azanyl-6-[(4-fluoro...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657132BDBM50657132(CHEMBL6102257)
Affinity DataEC50:  6.19E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657131BDBM50657131(CHEMBL6152617)
Affinity DataEC50:  7.61E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657122BDBM50657122(CHEMBL6152374)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657129BDBM50657129(CHEMBL6160920)
Affinity DataEC50:  9.39E+3nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657123BDBM50657123(CHEMBL6150201)
Affinity DataEC50:  1.01E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657112BDBM50657112(CHEMBL6160823)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657119BDBM50657119(CHEMBL6134168)
Affinity DataEC50:  1.27E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657133BDBM50657133(CHEMBL6133900)
Affinity DataEC50:  1.36E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657120BDBM50657120(CHEMBL6159804)
Affinity DataEC50:  1.36E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657114BDBM50657114(CHEMBL6120862)
Affinity DataEC50:  1.39E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657115BDBM50657115(CHEMBL6149068)
Affinity DataEC50:  1.84E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657130BDBM50657130(CHEMBL6145457)
Affinity DataEC50:  1.89E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657121BDBM50657121(CHEMBL6160237)
Affinity DataEC50:  3.03E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657134BDBM50657134(CHEMBL6168256)
Affinity DataEC50:  3.03E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657124BDBM50657124(CHEMBL6134101)
Affinity DataEC50:  3.53E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657118BDBM50657118(CHEMBL6143308)
Affinity DataEC50:  9.87E+4nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657125BDBM50657125(CHEMBL6146985)
Affinity DataEC50:  1.28E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657128BDBM50657128(CHEMBL6143038)
Affinity DataEC50:  1.31E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657117BDBM50657117(CHEMBL6133455)
Affinity DataEC50:  1.31E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657116BDBM50657116(CHEMBL6143850)
Affinity DataEC50:  1.64E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657127BDBM50657127(CHEMBL6152233)
Affinity DataEC50:  1.89E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657135BDBM50657135(CHEMBL6151567)
Affinity DataEC50:  1.96E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetVoltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3)(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657126BDBM50657126(CHEMBL6161725)
Affinity DataEC50:  2.18E+5nMAssay Description:Agonist activity at human KCNQ2/3 transfected in human HEK293 cells incubated for 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed