Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50023509
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at progesterone-induced progesterone receptor (unknown origin) transfected in human PC-3 cells by Dual Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at dexamethasone-induced glucocorticoid receptor (unknown origin) transfected in human PC-3 cells by Dual Luciferase reporter ass...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Antagonist activity at Androgen receptor F877L mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Antagonist activity at Androgen receptor F877L mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Antagonist activity at aldosterone-induced mineralocorticoid receptor (unknown origin) transfected in human PC-3 cells by Dual Luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 401nMAssay Description:Antagonist activity at Androgen receptor W742C mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 411nMAssay Description:Antagonist activity at Androgen receptor W742C mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 429nMAssay Description:Antagonist activity at Androgen receptor F877L/T878A mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Antagonist activity at LBP of Androgen receptor LBD (unknown origin) by PolarScreen competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 659nMAssay Description:Antagonist activity at Androgen receptor F877L/T878A mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 696nMAssay Description:Antagonist activity at Androgen receptor F877L/T878A mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 985nMAssay Description:Antagonist activity at Androgen receptor W742C mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at Androgen receptor F877L mutant expressed in human PC-3 cells co-expressing ARR2PB-luc by Dual-Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at LBP of Androgen receptor LBD (unknown origin) by PolarScreen competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.96E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.79E+3nMAssay Description:Antagonist activity at LBP of Androgen receptor LBD (unknown origin) by PolarScreen competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.53E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.64E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.53E+3nMAssay Description:Antagonist activity at LBP of Androgen receptor LBD (unknown origin) by PolarScreen competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.86E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.04E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at DHT-induced Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair















