Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50023010
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of OAT1 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Human)
Aligos Belgium BV
Curated by ChEMBL
Aligos Belgium BV
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of OAT3 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of AT1 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of MATE2 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of OCT1 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B3(Human)
Aligos Belgium BV
Curated by ChEMBL
Aligos Belgium BV
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of OATP1B3 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of MATE1 (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of BSEP (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Aligos Belgium BV
Curated by ChEMBL
Aligos Belgium BV
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of BCRP in human Caco-2 cells using estrone 3-sulfate as substrateMore data for this Ligand-Target Pair

