Compile Data Set for Download or QSAR
Report error Found 322 Enz. Inhib. hit(s) with all data for entry = 50023062
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658511BDBM50658511(CHEMBL6152639)
Affinity DataIC50: 1nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658478BDBM50658478(Camibirstat | Fhd-286)
Affinity DataIC50: 1nMAssay Description:Inhibition of BRG1 in human MDA-MB-231 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658488BDBM50658488(CHEMBL6133855)
Affinity DataIC50: 3nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658511BDBM50658511(CHEMBL6152639)
Affinity DataIC50: 3nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658488BDBM50658488(CHEMBL6133855)
Affinity DataIC50: 3nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658486BDBM50658486(CHEMBL6145659)
Affinity DataIC50: 4nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658485BDBM50658485(CHEMBL6164767)
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658484BDBM50658484(CHEMBL6166760)
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658483BDBM50658483(CHEMBL6168539)
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658485BDBM50658485(CHEMBL6164767)
Affinity DataIC50: 4nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658484BDBM50658484(CHEMBL6166760)
Affinity DataIC50: 4nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658486BDBM50658486(CHEMBL6145659)
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658511BDBM50658511(CHEMBL6152639)
Affinity DataIC50: 5nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658478BDBM50658478(Camibirstat | Fhd-286)
Affinity DataIC50: 5nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658516BDBM50658516(CHEMBL6162637)
Affinity DataIC50: 5nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658478BDBM50658478(Camibirstat | Fhd-286)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658510BDBM50658510(CHEMBL6141585)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658504BDBM50658504(CHEMBL6162908)
Affinity DataIC50: 6nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658520BDBM50658520(CHEMBL6167580)
Affinity DataIC50: 6nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658478BDBM50658478(Camibirstat | Fhd-286)
Affinity DataIC50: 6nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658517BDBM50658517(CHEMBL6144331)
Affinity DataIC50: 6nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658520BDBM50658520(CHEMBL6167580)
Affinity DataIC50: 6nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658510BDBM50658510(CHEMBL6141585)
Affinity DataIC50: 7nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658526BDBM50658526(CHEMBL6133150)
Affinity DataIC50: 7nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658520BDBM50658520(CHEMBL6167580)
Affinity DataIC50: 7nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658523BDBM50658523(CHEMBL6143779)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658517BDBM50658517(CHEMBL6144331)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658526BDBM50658526(CHEMBL6133150)
Affinity DataIC50: 9nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658510BDBM50658510(CHEMBL6141585)
Affinity DataIC50: 9nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658500BDBM50658500(CHEMBL6150430)
Affinity DataIC50: 9nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658507BDBM50658507(CHEMBL6171674)
Affinity DataIC50: 11nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658497BDBM50658497(CHEMBL6148030)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658504BDBM50658504(CHEMBL6162908)
Affinity DataIC50: 12nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658505BDBM50658505(CHEMBL6162601)
Affinity DataIC50: 13nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658499BDBM50658499(CHEMBL6149296)
Affinity DataIC50: 13nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658475BDBM50658475(CHEMBL6141925)
Affinity DataIC50: 14nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658521BDBM50658521(CHEMBL6145908)
Affinity DataIC50: 15nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658523BDBM50658523(CHEMBL6143779)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658526BDBM50658526(CHEMBL6133150)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658517BDBM50658517(CHEMBL6144331)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658486BDBM50658486(CHEMBL6145659)
Affinity DataIC50: 15nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658497BDBM50658497(CHEMBL6148030)
Affinity DataIC50: 18nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658475BDBM50658475(CHEMBL6141925)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658522BDBM50658522(CHEMBL6152455)
Affinity DataIC50: 20nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658495BDBM50658495(CHEMBL6149590)
Affinity DataIC50: 21nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658474BDBM50658474(CHEMBL6152213)
Affinity DataIC50: 21nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged BRM (unknown origin) (1 to 1590 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658510BDBM50658510(CHEMBL6141585)
Affinity DataIC50: 22nMAssay Description:Inhibition of BRG1 in human MDA-MB-231 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658507BDBM50658507(CHEMBL6171674)
Affinity DataIC50: 23nMAssay Description:Inhibition of C-terminal his6/FLAG-tagged BRG1 (unknown origin) (1 to 1647 residues) incubated for 2 hrs by ADP-glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658504BDBM50658504(CHEMBL6162908)
Affinity DataIC50: 23nMAssay Description:Inhibition of BRM in human A549 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Foghorn Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50658526BDBM50658526(CHEMBL6133150)
Affinity DataIC50: 25nMAssay Description:Inhibition of BRG1 in human MDA-MB-231 cells co-transfected with MMTV incubated for 6 hrs by bright-glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
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