Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50023114
TargetGABA-A receptor; alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50659308BDBM50659308(CHEMBL6163463)
Affinity DataEC50:  820nMAssay Description:Potentiation of recombinant human alpha1/beta2/gamma2 GABA receptor expressed in T-REX-CHO cells assessed as increase in current amplitude by whole-c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetGABA-A receptor; alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50659307BDBM50659307(CHEMBL6171514)
Affinity DataEC50:  1.24E+3nMAssay Description:Potentiation of recombinant human alpha1/beta2/gamma2 GABA receptor expressed in T-REX-CHO cells assessed as increase in current amplitude by whole-c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50659309BDBM50659309(CHEMBL6146779)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of Nav 1.2 (unknown origin) expressed in HEK293 cells at -20 mV to -120 mV holding potential under inactivation state by whole-cell patch ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50659307BDBM50659307(CHEMBL6171514)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Nav 1.2 (unknown origin) expressed in HEK293 cells at -20 mV to -120 mV holding potential under inactivation state by whole-cell patch ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed