Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50023161
Affinity DataKd: 6nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 22nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 80nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 80nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 180nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataEC50: 244nMAssay Description:Inhibition of CypD mediated opening to mitochondrial transition pore in human HepG2 cells by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 360nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataEC50: 463nMAssay Description:Inhibition of CypD mediated opening to mitochondrial transition pore in human HepG2 cells by FLIPR analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 580nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding affinity to human CypA assessed as dissociation constant by SPR methodMore data for this Ligand-Target Pair
Affinity DataKd: 670nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 960nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 1.01E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 1.16E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 2.40E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 2.97E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 4.60E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 5.70E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 5.85E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 6.30E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 7.10E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: 8.75E+3nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: 9.10E+3nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypA (1 to 165 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation c...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase F, mitochondrial(Human)
University of Edinburgh
Curated by ChEMBL
University of Edinburgh
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human full length N-terminal CypD (42 to 207 residues) extracted from Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair



















