Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50023231
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Displacement of fluorophore-labeled probe from TYK2 JH2 domain (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Displacement of fluorophore-labeled probe from TYK2 JH2 domain (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Displacement of fluorophore-labeled probe from TYK2 JH2 domain (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of fluorophore-labeled probe from JAK1 JH2 domain (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of fluorophore-labeled probe from JAK1 JH2 domain (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to JAK3 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to JAK2 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to JAK1 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to TYK2 JH1 domain (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair


