Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50023799
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of recombinant human PIM-1 extracted from bacteria using histone H1 as substrate incubated for 30 mins in presence of ATP by ADP-Glo kinas...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite Clermont Auvergne
Curated by ChEMBL
Universite Clermont Auvergne
Curated by ChEMBL
Affinity DataIC50: 159nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) extracted from bacteria using KKISGRLSPIMTEQ as substrate incubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 173nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant mouse CLK1 extracted from bacteria using GRSRSRSRSRSR as substrate incubated for 30 mins in presence of ATP by ADP-Glo kina...More data for this Ligand-Target Pair
Affinity DataIC50: 237nMAssay Description:Inhibition of recombinant mouse CLK1 extracted from bacteria using GRSRSRSRSRSR as substrate incubated for 30 mins in presence of ATP by ADP-Glo kina...More data for this Ligand-Target Pair
Affinity DataIC50: 258nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) extracted from bacteria using histone H3 (1 to 21) peptide as substrate in...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite Clermont Auvergne
Curated by ChEMBL
Universite Clermont Auvergne
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) extracted from bacteria using KKISGRLSPIMTEQ as substrate incubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 387nMAssay Description:Inhibition of recombinant mouse CLK1 extracted from bacteria using GRSRSRSRSRSR as substrate incubated for 30 mins in presence of ATP by ADP-Glo kina...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite Clermont Auvergne
Curated by ChEMBL
Universite Clermont Auvergne
Curated by ChEMBL
Affinity DataIC50: 498nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) extracted from bacteria using KKISGRLSPIMTEQ as substrate incubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 546nMAssay Description:Inhibition of recombinant mouse CLK1 extracted from bacteria using GRSRSRSRSRSR as substrate incubated for 30 mins in presence of ATP by ADP-Glo kina...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite Clermont Auvergne
Curated by ChEMBL
Universite Clermont Auvergne
Curated by ChEMBL
Affinity DataIC50: 602nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) extracted from bacteria using KKISGRLSPIMTEQ as substrate incubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 876nMAssay Description:Inhibition of recombinant human PIM-1 extracted from bacteria using histone H1 as substrate incubated for 30 mins in presence of ATP by ADP-Glo kinas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of recombinant human PIM-1 extracted from bacteria using histone H1 as substrate incubated for 30 mins in presence of ATP by ADP-Glo kinas...More data for this Ligand-Target Pair
