Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50023600
Affinity DataKd: 0.0580nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.0600nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.160nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.220nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.25nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.280nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 0.630nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 4.60nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Inverse agonist activity at N-terminal his-tagged wild type human RORgammat LBD domain expressed in Escherichia coli assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at RORgammat in mouse whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17A production incubated for 1 hrs by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+3nMAssay Description:Inverse agonist activity at human RORgammat by mammalian 1-hybrid assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.20E+3nMAssay Description:Inverse agonist activity at human RORbeta assessed as dissociation constant by thermofluor assayMore data for this Ligand-Target Pair

















