Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50023601
Affinity DataKi: 1.90nMAssay Description:Competitive inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed a inhibition cons...More data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Binding affinity to laforin (unknown origin) assessed as dissociation constant by MST analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Competitive inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed a inhibition cons...More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 131nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 glucan phosphatase activity using amylopectin as substrate by ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 261nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 289nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 3.14E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 4.05E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 4.72E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 9.33E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 9.87E+3nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
Affinity DataKi: 2.47E+4nMAssay Description:Competitive inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed a inhibition cons...More data for this Ligand-Target Pair
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of His-tagged SHP2 (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotometr...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged laforin (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate assessed as substrate hydrolysis incub...More data for this Ligand-Target Pair
TargetLow molecular weight phosphotyrosine protein phosphatase(Human)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged LMW-PTP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotom...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase delta(Homo sapiens)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged PTP-delta (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophot...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged Yersinia pseudotuberculosis IP32953 YopH extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged Yersinia pseudotuberculosis IP32953 YopH extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins ...More data for this Ligand-Target Pair
TargetLow molecular weight phosphotyrosine protein phosphatase(Human)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged LMW-PTP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotom...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged TC-PTP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged PTP-alpha (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophot...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged PTP-alpha (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophot...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged PTP-beta (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophoto...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged HePTP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged STEP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotometr...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged STEP (unknown origin) extracted from Escherichia coli BL21 using pNPP as substrate incubated for 80 mins by spectrophotometr...More data for this Ligand-Target Pair




























