Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50023602
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal hexahistidine-tagged human PARP14 (1611 to 1801 residues) catalytic domain extracted from Escherichia coli BL21-CodonPlus (D...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.20nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of fluorescently-labeled PARP14 (unknown origin) by small molecule microarray based analysisMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP15(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 916nMAssay Description:Inhibition of PARP15 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP12(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of PARP12 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of PARP5b (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of PARP5a (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of PARP7 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of PARP3 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP11(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.75E+3nMAssay Description:Inhibition of PARP11 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.23E+3nMAssay Description:Inhibition of PARP10 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
























3D Structure (crystal)