Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50023271
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661232BDBM50661232(CHEMBL6171555)
Affinity DataIC50: 41nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661236BDBM50661236(CHEMBL6142609)
Affinity DataIC50: 48nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661236BDBM50661236(CHEMBL6142609)
Affinity DataIC50: 70nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661232BDBM50661232(CHEMBL6171555)
Affinity DataIC50: 78nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661233BDBM50661233(CHEMBL6170224)
Affinity DataIC50: 79nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661237BDBM50661237(CHEMBL6168079)
Affinity DataIC50: 81nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 92nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661237BDBM50661237(CHEMBL6168079)
Affinity DataIC50: 109nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661233BDBM50661233(CHEMBL6170224)
Affinity DataIC50: 119nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 147nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661239BDBM50661239(CHEMBL6163498)
Affinity DataIC50: 165nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661239BDBM50661239(CHEMBL6163498)
Affinity DataIC50: 165nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661235BDBM50661235(CHEMBL6120511)
Affinity DataIC50: 174nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661235BDBM50661235(CHEMBL6120511)
Affinity DataIC50: 231nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661238BDBM50661238(CHEMBL6174125)
Affinity DataIC50: 450nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661234BDBM50661234(CHEMBL6148739)
Affinity DataIC50: 459nMAssay Description:Inhibition of human DYRK1A using DYTKtide as substrate incubated for 60 mins in presence of ATP by ADP-gloreagent based multimode reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661238BDBM50661238(CHEMBL6174125)
Affinity DataIC50: 566nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Instituto de Ciencias Matemeticas (ICMAT-CSIC)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661234BDBM50661234(CHEMBL6148739)
Affinity DataIC50: 577nMAssay Description:Inhibition of full length recombinant human DYRK1B expressed in baculovirus in Sf9 insect cells using RRRFRPASPLRGPPK as substrate incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed