| Assay Method Information | |
| | ChEMBL_2640794 |
| Description: | Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed inhibition of epibatidine-induced calcium flux preincubated for 10 mins followed by epibatidine addition by FLIPR Calcium-6 assay |
| Affinity data for this assay | |
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